Pharmacokinetic | Unit | Free-TGC | CSs-TGC | Aβ11/T80@CSs-TGC |
---|---|---|---|---|
Cmax | μg/mL | 3.70 ± 0.62 | 8.09 ± 0.35** | 10.72 ± 2.26*** |
Tmax | h | 0.25 | 0.25 | 0.25 |
AUC(0-t) | μg/mL*h | 8.48 ± 2.90 | 16.51 ± 0.09* | 21.62 ± 1.79** |
T1/2 | h | 0.77 ± 0.24 | 0.91 ± 0.21 | 1.26 ± 0.21 |
MRT(0-t) | h | 2.6 ± 0.16 | 2.29 ± 0.10 | 2.39 ± 0.14 |
CL | L/h/kg | 1.20 ± 0.25 | 0.59 ± 0.03 | 0.43 ± 0.02 |